Bromide

Bromide

SCHEMBL29831731

Br.Cc1ccc(S(=O)(=O)N(C)[C@@H](Cc2ccccn2)C(=O)O)cc1

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 known ✓ P07550 1/20 0.43
ADAMTS5 Q9UNA0 1/20 0.51
KMT2A Q03164 5/20 0.48
MEN1 O00255 1/20 0.48
PTPRA P18433 1/20 0.46
GAA P10253 1/20 0.46
ALDH1A1 P00352 2/20 0.45
CYP3A4 P08684 1/20 0.45
KDM4E B2RXH2 3/20 0.45
POLB P06746 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.43
MAPT P10636 1/20 0.43
HSD17B10 Q99714 1/20 0.43
PTGS2 P35354 1/20 0.43
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
AGER Q15109 1/20 0.42
NPC1 O15118 1/20 0.41
TP53 P04637 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16058321 0.99 ADAMTS5 (0.52) ADAMTS5KMT2AMEN1PTPRAGAA
SCHEMBL21885547 0.99 ADAMTS5 (0.52) ADAMTS5KMT2AMEN1PTPRAGAA
SCHEMBL5573300 0.81 ADAMTS5 (0.73) ADAMTS5KMT2AGAAPOLBMAPT
SCHEMBL5573297 0.81 ADAMTS5 (0.73) ADAMTS5KMT2AGAAPOLBMAPT
SCHEMBL28583121 0.79 MEN1 (0.48) ADAMTS5KMT2AMEN1PTPRAGAA
SCHEMBL5572738 0.76 GAA (0.59) KMT2AMEN1GAAALDH1A1CYP3A4
SCHEMBL17481680 0.76 AGER (0.54) ADAMTS5KMT2AMEN1ALDH1A1MAPT
SCHEMBL5573156 0.76 AGER (0.54) ADAMTS5KMT2AALDH1A1MAPTKEAP1
SCHEMBL21885546 0.74 TDP1 (0.58) ADAMTS5KMT2AALDH1A1POLBMAPT
SCHEMBL18858366 0.74 PTPRA (0.48) KMT2AMEN1PTPRAALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110016020-B Compound or pharmaceutically acceptable salt thereof, application and pharmaceutical composition thereof 赛克里翁治疗有限公司 2022-07-26 CN disclosed