SCHEMBL29907667

SCHEMBL29907667

NC(=O)c1cnc(-c2ccc[nH]2)cn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.49
SIRT6 Q8N6T7 2/20 0.44
PARP1 P09874 1/20 0.43
GSK3B P49841 1/20 0.42
KDR P35968 1/20 0.42
ADORA3 P0DMS8 1/20 0.38
TSHR P16473 1/20 0.38
MC4R P32245 1/20 0.38
ADRA1A P35348 1/20 0.38
MC3R P41968 1/20 0.38
KMT2A Q03164 1/20 0.37
IKBKE Q14164 1/20 0.36
TBK1 Q9UHD2 1/20 0.36
MAPK1 P28482 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HPGDS O60760 1/20 0.34
TGFBR1 P36897 1/20 0.34
LCK P06239 1/20 0.33
CSNK1A1 P48729 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12248222 0.88 KDM4C (0.54) KDM4CPARP1KDRTSHRKMT2A
SCHEMBL2933552 0.74 LDHA (0.53) SIRT6GSK3BTSHRMAPK1
SCHEMBL20852324 0.73 NPC1 (0.58) KDRKMT2AIKBKETBK1
SCHEMBL2635320 0.73 SIRT6 (0.73) SIRT6GSK3BADORA3TSHRMC4R
SCHEMBL27646753 0.71 P4HTM (0.49) KDM4CSIRT6GSK3BADORA3TSHR
SCHEMBL3868273 0.71 P4HA1 (0.63) KDM4CPARP1KDRHDAC1HDAC6
SCHEMBL30968251 0.71 KDM4C (0.47) KDM4CPARP1IKBKETBK1HDAC1
Hydrochloric Acid SCHEMBL27917292 0.71 SIRT6 (0.70) SIRT6GSK3BADORA3TSHRMC4R
SCHEMBL28045606 0.70 SIRT6 (0.44) SIRT6GSK3BADORA3TSHRMC4R
SCHEMBL7942874 0.69 KDM4C (0.40) KDM4CPARP1KDRADRA1AHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115181092-A Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-10-14 CN disclosed
CN-112279837-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-08-09 CN disclosed