SCHEMBL28045606

SCHEMBL28045606

NC(=O)c1cnc(-c2c(F)cccc2F)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 2/20 0.44
DHODH Q02127 1/20 0.40
HPGDS O60760 1/20 0.40
KMT2A Q03164 1/20 0.40
PIM1 P11309 1/20 0.40
PIM3 Q86V86 1/20 0.40
TGFBR1 P36897 2/20 0.39
GSK3B P49841 1/20 0.39
ALOX5AP P20292 2/20 0.39
FEN1 P39748 2/20 0.39
CA5A P35218 1/20 0.39
TTR P02766 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
TSHR P16473 1/20 0.38
MC4R P32245 1/20 0.38
ADRA1A P35348 1/20 0.38
MC3R P41968 1/20 0.38
GRM2 Q14416 1/20 0.37
HTR5A P47898 1/20 0.36
SCN9A Q15858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29551864 0.78 HPGDS (0.63) SIRT6DHODHHPGDSPIM1PIM3
SCHEMBL29907612 0.75 NPC1 (0.50) SIRT6HPGDSKMT2APIM1PIM3
SCHEMBL2933552 0.74 LDHA (0.53) SIRT6GSK3BTSHR
SCHEMBL2635320 0.73 SIRT6 (0.73) SIRT6KMT2AGSK3BADORA3TSHR
SCHEMBL4651415 0.72 P4HA1 (0.66) DHODHHPGDSTTRNPC1P4HTM
SCHEMBL379465 0.71 LDHA (0.47) SIRT6HPGDSKMT2AGSK3BALOX5AP
SCHEMBL27646753 0.71 P4HTM (0.49) SIRT6HPGDSKMT2ATGFBR1GSK3B
Hydrochloric Acid SCHEMBL27917292 0.71 SIRT6 (0.70) SIRT6KMT2AGSK3BADORA3TSHR
SCHEMBL29907667 0.70 KDM4C (0.49) SIRT6HPGDSKMT2ATGFBR1GSK3B
SCHEMBL29600561 0.70 ATR (0.52) PIM1PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105566311-A Oxazole and isoxazole crac modulators LUPIN LTD 2016-05-11 CN disclosed
CN-103228636-B Calcium modulators of oxazole and isoxazole calcium release activation LUPIN LTD. (IN) 2016-02-10 CN disclosed