SCHEMBL29910078

SCHEMBL29910078

O=C1c2ccccc2C(=O)N1Cc1nnc(Cl)cc1N1CC2CCCC2C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.40
HTR7 P34969 1/20 0.40
HRH1 P35367 1/20 0.40
DRD3 P35462 1/20 0.40
HTR2B P41595 1/20 0.40
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
GRM5 P41594 1/20 0.37
MAPT P10636 2/20 0.36
RECQL P46063 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
HTT P42858 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
ADRA1D P25100 2/20 0.36
ADRA1A P35348 2/20 0.36
ADRA1B P35368 2/20 0.36
TYR P14679 2/20 0.35
CASP3 P42574 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24941131 1.00 HTR1A (0.40) HTR1AHTR7HRH1DRD3HTR2B
SCHEMBL24941127 0.77 SMPD3 (0.30)
SCHEMBL24941130 0.76
SCHEMBL28846456 0.74 MAPK1 (0.46) ALDH1A1KDM4EGRM5MAPTRECQL
SCHEMBL29893702 0.74 MAPK1 (0.46) ALDH1A1KDM4EGRM5MAPTRECQL
SCHEMBL24941129 0.74
SCHEMBL21555613 0.67 TYR (0.46) ALDH1A1GRM5MAPTRECQLCYP1A2
SCHEMBL28846377 0.65 HTR3A (0.36)
SCHEMBL399990 0.64 ALDH1A1 (0.54) ALDH1A1KDM4EGRM5MAPTRECQL
SCHEMBL24719019 0.64 ALDH1A1 (0.54) ALDH1A1KDM4EMAPTRECQLCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055026-A1 COMPOUNDS AS CD73 INHIBITORS Bioardis LLC (US) 2022-09-14 EP disclosed