SCHEMBL29923210

SCHEMBL29923210

CCOC(=O)c1cc(CC)cc2c(Br)cc(C)nc12

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
CYP4F2 P78329 1/20 0.41
CYP4A11 Q02928 1/20 0.41
KDM4E B2RXH2 5/20 0.40
KMT2A Q03164 3/20 0.40
TSHR P16473 2/20 0.40
MEN1 O00255 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB2 P47870 1/20 0.40
ATM Q13315 1/20 0.39
MAPT P10636 2/20 0.39
MAOB P27338 1/20 0.38
IKBKB O14920 1/20 0.38
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24915691 1.00 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2L3MBTL1CYP4F2CYP4A11
SCHEMBL29923655 0.84 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2L3MBTL1KDM4EKMT2A
SCHEMBL24916324 0.84 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2L3MBTL1KDM4EKMT2A
SCHEMBL24916059 0.82 POLB (0.41) ALDH1A1SMN1; SMN2L3MBTL1CYP4F2CYP4A11
SCHEMBL29923420 0.81 GABRA1 (0.45) ALDH1A1SMN1; SMN2CYP4F2CYP4A11KDM4E
SCHEMBL22750311 0.81 GABRA1 (0.45) ALDH1A1SMN1; SMN2CYP4F2CYP4A11KDM4E
SCHEMBL3928069 0.74 CA12 (0.43) ALDH1A1SMN1; SMN2L3MBTL1CYP4F2CYP4A11
SCHEMBL6586612 0.73 CCR6 (0.53) ALDH1A1SMN1; SMN2L3MBTL1KDM4EKMT2A
SCHEMBL22766603 0.72 GABRA1 (0.47) ALDH1A1SMN1; SMN2L3MBTL1CYP4F2CYP4A11
SCHEMBL24916110 0.71 CA12 (0.47) ALDH1A1CYP4F2CYP4A11KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed