SCHEMBL29923655

SCHEMBL29923655

CCOC(=O)c1cc(OC)cc2c(Br)cc(C)nc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.44
KDM4E B2RXH2 6/20 0.44
HPGD P15428 5/20 0.44
DPP4 P27487 2/20 0.44
CDC25B P30305 1/20 0.42
CYP3A4 P08684 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
MAOB P27338 2/20 0.40
CA12 O43570 1/20 0.40
CA2 P00918 1/20 0.40
GLA P06280 1/20 0.40
CA3 P07451 1/20 0.40
GAA P10253 1/20 0.40
CA4 P22748 1/20 0.40
CA6 P23280 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24916324 1.00 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDDPP4CDC25B
SCHEMBL29923598 0.86 HPGD (0.48) ALDH1A1KDM4EHPGDDPP4CDC25B
SCHEMBL29923210 0.84 ALDH1A1 (0.42) ALDH1A1KDM4ESMN1; SMN2L3MBTL1MAOB
SCHEMBL24915691 0.84 ALDH1A1 (0.42) ALDH1A1KDM4ESMN1; SMN2L3MBTL1MAOB
SCHEMBL24915919 0.82 HPGD (0.43) ALDH1A1KDM4EHPGDDPP4CDC25B
SCHEMBL24915732 0.82 DPP4 (0.46) ALDH1A1KDM4EHPGDDPP4CDC25B
SCHEMBL29923458 0.82 DPP4 (0.46) ALDH1A1KDM4EHPGDDPP4CDC25B
SCHEMBL19783054 0.74 HPGD (0.48) ALDH1A1KDM4EHPGDDPP4CDC25B
SCHEMBL22750299 0.73 CRHR1 (0.47) ALDH1A1CYP3A4SMN1; SMN2GAAPOLB
SCHEMBL29923906 0.73 CRHR1 (0.47) ALDH1A1CYP3A4SMN1; SMN2GAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed