SCHEMBL29923722

SCHEMBL29923722

CCc1ccc2c(c1)C=CCN2C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.38
TRPA1 O75762 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2A6 P11509 1/20 0.33
GABRA1 P14867 4/20 0.33
GABRA5 P31644 4/20 0.33
SRD5A1 P18405 1/20 0.33
MGLL Q99685 3/20 0.31
GABRG2 P18507 3/20 0.31
GABRB3 P28472 3/20 0.31
GABRA3 P34903 3/20 0.31
GABRA2 P47869 3/20 0.31
GABRA6 Q16445 3/20 0.31
GABRB2 P47870 2/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29923614 0.76 HTR2C (0.38) BRD4
SCHEMBL30847749 0.76 HSD11B1 (0.40) ALDH1A1MAPT
SCHEMBL23346796 0.74 MAPT (0.39) SLC6A2SLC6A4ALDH1A1LMNAMAPT
SCHEMBL14283937 0.74 ESR1 (0.35) CYP1A2LMNAMAPT
SCHEMBL5714026 0.74 SRD5A1 (0.35) BRD4TRPA1CYP1A2CYP2A6GABRA1
Iodide SCHEMBL28915713 0.73 HSD17B3 (0.40) SLC6A3ALDH1A1LMNAMAPK1SMN1; SMN2
Hydrochloric Acid SCHEMBL28747930 0.73 MAPT (0.41) SLC6A2SLC6A4ALDH1A1LMNAMAPT
SCHEMBL28599880 0.71 ALDH1A1 (0.36) ALDH1A1MAPTMAPK1L3MBTL1
SCHEMBL10670398 0.70 CA12 (0.34) BRD4SRD5A1SLC6A3NPC1MAPT
Iodide SCHEMBL30293255 0.70 LMNA (0.39) BRD4CYP1A2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed