SCHEMBL29930814

SCHEMBL29930814

C[Si](C)(C)CCOCn1ncc2cc(-c3ccsc3)cnc21

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 10/20 0.41
PDGFRA P16234 10/20 0.41
KDR P35968 4/20 0.39
CYP2A6 P11509 3/20 0.38
FLT1 P17948 2/20 0.36
FLT4 P35916 2/20 0.36
GAK O14976 1/20 0.36
CHEK2 O96017 1/20 0.35
DGAT1 O75907 1/20 0.35
CYP2E1 P05181 1/20 0.35
CYP2B6 P20813 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29930600 0.81 HDAC8 (0.36) DGAT1
SCHEMBL29930403 0.81 FTO (0.39) DGAT1
SCHEMBL29930423 0.79 MAP4K4 (0.40) DGAT1
SCHEMBL31469272 0.78 DGAT1 (0.35) DGAT1
SCHEMBL29930774 0.78 DGAT1 (0.41) GAKDGAT1
SCHEMBL29930433 0.78 DGAT1 (0.41) PDGFRBPDGFRADGAT1
SCHEMBL1565921 0.76 DGAT1 (0.40) DGAT1
SCHEMBL29705469 0.76 DGAT1 (0.33) DGAT1
SCHEMBL18188139 0.76 DGAT1 (0.33) DGAT1
SCHEMBL19023260 0.76 DGAT1 (0.33) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022235097-A1 PHARMACEUTICAL COMPOSITION CONTAINING NOVEL PYRAZOLO[3,4-B]PYRIDINE DERIVATIVE FOR PREVENTION OR TREATMENT OF METABOLIC DISEASE INCLUDING OBESITY AND DIABETES MELLITUS OR NONALCOHOLIC STEATOHEPATITIS 한국화학연구원 2022-11-10 WO disclosed