SCHEMBL29930600

SCHEMBL29930600

C[Si](C)(C)CCOCn1ncc2cc(-c3cncnc3)cnc21

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.36
DGAT1 O75907 6/20 0.35
MAPT P10636 1/20 0.33
CHRNB1 P11230 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNB3 Q05901 1/20 0.31
ALOX5AP P20292 1/20 0.30
FEN1 P39748 1/20 0.30
BRD4 O60885 1/20 0.30
CREBBP Q92793 1/20 0.30
F2RL1 P55085 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29930403 0.87 FTO (0.39) DGAT1MAPTALOX5APFEN1BRD4
SCHEMBL29930814 0.81 PDGFRB (0.41) DGAT1
SCHEMBL29930423 0.81 MAP4K4 (0.40) DGAT1CHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL18188139 0.80 DGAT1 (0.33) DGAT1ALOX5APFEN1F2RL1
SCHEMBL19023260 0.80 DGAT1 (0.33) DGAT1MAPTF2RL1
SCHEMBL29705469 0.80 DGAT1 (0.33) DGAT1MAPTF2RL1
SCHEMBL1565921 0.80 DGAT1 (0.40) HDAC8DGAT1F2RL1
SCHEMBL31469272 0.79 DGAT1 (0.35) DGAT1MAPTALOX5APFEN1BRD4
SCHEMBL29930774 0.79 DGAT1 (0.41) DGAT1ALOX5APFEN1BRD4CREBBP
SCHEMBL29705384 0.79 HPGDS (0.36) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022235097-A1 PHARMACEUTICAL COMPOSITION CONTAINING NOVEL PYRAZOLO[3,4-B]PYRIDINE DERIVATIVE FOR PREVENTION OR TREATMENT OF METABOLIC DISEASE INCLUDING OBESITY AND DIABETES MELLITUS OR NONALCOHOLIC STEATOHEPATITIS 한국화학연구원 2022-11-10 WO disclosed