SCHEMBL29934305

SCHEMBL29934305

O=C1C=CC(=O)N1Nc1cccc(-c2cccc(C(F)(F)F)c2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.48
CTSS P25774 1/20 0.48
XPO1 O14980 1/20 0.47
KMO O15229 2/20 0.44
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
CNR2 P34972 2/20 0.42
CNR1 P21554 1/20 0.42
MAOB P27338 1/20 0.41
KARS1 Q15046 2/20 0.41
IDO1 P14902 1/20 0.41
LMNA P02545 1/20 0.40
KDR P35968 1/20 0.40
EPHB4 P54760 1/20 0.40
KDM1A O60341 2/20 0.40
ADORA2A P29274 1/20 0.40
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29934354 0.85 XPO1 (0.47) XDHCTSSXPO1KMOKDM4E
SCHEMBL1592508 0.85 XPO1 (0.47) XDHCTSSXPO1KMOKDM4E
SCHEMBL1592510 0.84 XDH (0.45) XDHCTSSKMOKDM4EALDH1A1
SCHEMBL30346302 0.68 XPO1 (0.63) XDHXPO1ADORA2A
SCHEMBL4787 0.68 CTSS (0.60) XDHCTSSKMOKDM4EALDH1A1
SCHEMBL6256565 0.68 CTSS (0.60) XDHCTSSKMOKDM4EALDH1A1
SCHEMBL2615262 0.68 CTSS (0.60) XDHCTSSKMOKDM4EALDH1A1
SCHEMBL3999574 0.68 CTSS (0.60) XDHCTSSKMOKDM4EALDH1A1
SCHEMBL2304614 0.68 CTSS (0.56) XDHCTSSKMOKDM4EALDH1A1
SCHEMBL14152109 0.67 KMO (0.66) XDHCTSSKMOKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4074704-A1 QUINOLINE COMPOUNDS WITH ANTI-CANCER ACTIVITY CanBas Co., Ltd. (JP) 2022-10-19 EP disclosed