SCHEMBL29937403

SCHEMBL29937403

C#Cc1nc([Si](C(C)C)(C(C)C)C(C)C)cc2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.31
CYP2A6 P11509 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HIF1A Q16665 1/20 0.31
CYP1B1 Q16678 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL648767 0.69
SCHEMBL15940607 0.68 ADORA3 (0.44) ALDH1A1
SCHEMBL29977359 0.68 TRPM4 (0.33) ALDH1A1
SCHEMBL27770259 0.65 ALDH1A1 (0.32) ALDH1A1HIF1ACYP1B1HSD17B10
SCHEMBL2418686 0.62 CYP2A6 (0.50) CYP1A2CYP2A6ALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL27779935 0.61 NCF1 (0.33) CYP1A2CYP2A6ALDH1A1HIF1ACYP1B1
SCHEMBL12278288 0.61 HPRT1 (0.50) CYP1A2CYP2A6ALDH1A1HIF1ACYP1B1
SCHEMBL12405251 0.61 HPRT1 (0.50) CYP1A2CYP2A6ALDH1A1HIF1ACYP1B1
SCHEMBL4572766 0.60 GABRP (0.33) CYP1A2ALDH1A1
SCHEMBL738593 0.60 ALDH1A1 (0.44) CYP1A2CYP2A6ALDH1A1HIF1ACYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4322954-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT Merck Sharp & Dohme LLC (US) 2024-02-21 EP disclosed
WO-2022221739-A1 SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT MERCK SHARP & DOHME CORP. (US) 2022-10-20 WO disclosed