SCHEMBL29950001

SCHEMBL29950001

O=c1oc(=O)n(CC2CCN(c3ccccc3Cl)CC2)c2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
GRM2 Q14416 1/20 0.42
HSD11B1 P28845 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29949593 0.84 HTR1A (0.44)
SCHEMBL5259729 0.84 DHFR (0.46) TSHR
SCHEMBL6689039 0.81 NPC1 (0.45) TSHR
SCHEMBL5260181 0.80 NPC1 (0.50)
SCHEMBL1716008 0.79 CNR2 (0.48)
SCHEMBL6737897 0.74 CNR2 (0.46) TSHR
SCHEMBL28849138 0.72 GSK3B (0.52)
SCHEMBL29950200 0.72 GSK3B (0.52)
SCHEMBL3580000 0.71 NOS3 (0.44)
SCHEMBL6235260 0.71 TSHR (0.63) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108069952-B Quinolinone compound and application thereof in medicines 广东东阳光药业有限公司 2022-09-27 CN disclosed