SCHEMBL29951490

SCHEMBL29951490

CCc1ccc(-c2[nH]c3cc(F)cc(F)c3c2C=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.43
PARP2 Q9UGN5 6/20 0.40
DYRK3 O43781 1/20 0.39
TNKS O95271 1/20 0.39
PGR P06401 1/20 0.39
CDK1 P06493 1/20 0.39
ADRB1 P08588 1/20 0.39
POLA1 P09884 1/20 0.39
PIM1 P11309 1/20 0.39
SLC6A2 P23975 1/20 0.39
ADRA1A P35348 1/20 0.39
PTGS2 P35354 1/20 0.39
CDK16 Q00536 1/20 0.39
PDE4D Q08499 1/20 0.39
KCNH2 Q12809 1/20 0.39
DYRK1A Q13627 1/20 0.39
PARP15 Q460N3 1/20 0.39
PARP14 Q460N5 1/20 0.39
PARP10 Q53GL7 1/20 0.39
PIM3 Q86V86 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29953952 0.86 KDM4E (0.37) PARP1PTGS2TNKS2MAPK14CTSV
SCHEMBL29955797 0.85 KDM4E (0.38) PARP1PARP2DYRK3TNKSPGR
SCHEMBL15331672 0.83 PARP1 (0.36) PARP1PTGS2PARP3GCGRMAPK14
SCHEMBL15331326 0.82 MAPK13 (0.38) PARP1PARP2DYRK3TNKSPGR
SCHEMBL2559858 0.82 GPR17 (0.35) PARP1GPR17
SCHEMBL2559831 0.81 PTGS2 (0.34) PARP1PGRPTGS2PARP3GPR17
SCHEMBL29952478 0.80 APOL1 (0.44)
SCHEMBL29958306 0.78 ERN1 (0.38) PARP1CTSVCTSLGPR17
SCHEMBL2558994 0.78 PTGS2 (0.44) PTGS2GCGRMAPK14CTSVCTSL
SCHEMBL29957654 0.77 ALDH1A1 (0.39) TNKS2MAPK14LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed