SCHEMBL29954099

SCHEMBL29954099

CCN(CC(=O)NC)c1ccc(C=O)cc1C

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A3 P47895 5/20 0.49
ALDH3A1 P30838 5/20 0.45
ALDH1A1 P00352 11/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CRHR1 P34998 1/20 0.36
CYP2A6 P11509 1/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 2/20 0.33
GAA P10253 2/20 0.33
GFER P55789 2/20 0.33
POLB P06746 1/20 0.33
GLA P06280 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2560265 0.89 ALDH1A1 (0.51) ALDH1A3ALDH3A1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL29951697 0.88 ALDH1A3 (0.48) ALDH1A3ALDH3A1ALDH1A1SMN1; SMN2HPGD
SCHEMBL2555933 0.86 ALDH1A1 (0.44) ALDH1A3ALDH3A1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL29951185 0.85 ALDH1A3 (0.46) ALDH1A3ALDH3A1ALDH1A1KDM4EGAA
SCHEMBL29953881 0.85 ALDH1A3 (0.48) ALDH1A3ALDH3A1ALDH1A1SMN1; SMN2POLB
SCHEMBL9362085 0.83 ALDH1A3 (0.67) ALDH1A3ALDH3A1ALDH1A1CYP2A6MAPT
SCHEMBL29950930 0.81 ALDH3A1 (0.74) ALDH1A3ALDH3A1ALDH1A1SMN1; SMN2MAPT
SCHEMBL29952860 0.79 ALDH1A1 (0.65) ALDH1A3ALDH3A1ALDH1A1SMN1; SMN2CYP2A6
SCHEMBL29953969 0.77 ALDH1A3 (0.43) ALDH1A3ALDH3A1ALDH1A1CYP2A6KDM4E
SCHEMBL24833805 0.76 LMNA (0.45) ALDH1A1MAPTKDM4EGAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed