SCHEMBL29957448

SCHEMBL29957448

O=Cc1c(C2CC2)[nH]c2ccc(Br)cc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.42
PIM1 P11309 2/20 0.42
PIM3 Q86V86 1/20 0.42
DHODH Q02127 1/20 0.41
LMNA P02545 2/20 0.40
HPGD P15428 1/20 0.40
MAPT P10636 3/20 0.39
KCNH2 Q12809 1/20 0.39
GSK3B P49841 3/20 0.39
SIRT1 Q96EB6 1/20 0.39
ALDH1A1 P00352 2/20 0.38
HSD17B10 Q99714 1/20 0.38
MAPK1 P28482 1/20 0.38
MAPKAPK2 P49137 1/20 0.38
SLC6A4 P31645 2/20 0.37
CHEK1 O14757 1/20 0.37
AURKA O14965 1/20 0.37
DAPK3 O43293 1/20 0.37
JAK2 O60674 1/20 0.37
PRKD3 O94806 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29957067 0.82 SIRT1 (0.45) LMNAHPGDMAPTSIRT1ALDH1A1
SCHEMBL29956270 0.78 KDM4E (0.44) GSK3BCDK5CHUK
SCHEMBL15332502 0.78 KDM4E (0.42) MAPTALDH1A1HTT
SCHEMBL15330972 0.78 KIF11 (0.44) MAPT
SCHEMBL3223692 0.78 ALDH1A1 (0.50) HPGDMAPTSIRT1ALDH1A1HSD17B10
SCHEMBL29957756 0.78 ALDH1A1 (0.50) HPGDMAPTSIRT1ALDH1A1HSD17B10
SCHEMBL7254612 0.78 AHR (0.43) HPGDMAPTGSK3BSIRT1ALDH1A1
SCHEMBL29952591 0.77 MAPT (0.52) LMNAMAPTALDH1A1HTT
SCHEMBL29957489 0.75 SIRT1 (0.46) LMNAHPGDMAPTSIRT1ALDH1A1
SCHEMBL29953259 0.75 KDM4E (0.48) HPGDMAPTALDH1A1HSD17B10MAPKAPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed