SCHEMBL29967361

SCHEMBL29967361

S=c1[nH]c2ncccc2s1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB8 P28062 8/20 0.50
KDM4E B2RXH2 4/20 0.50
ALDH1A1 P00352 4/20 0.50
HPGD P15428 2/20 0.50
CYP3A4 P08684 1/20 0.50
ALOX15 P16050 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
HTT P42858 1/20 0.44
HSD17B10 Q99714 1/20 0.44
GAA P10253 2/20 0.37
MAPT P10636 2/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
GFER P55789 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
AXL P30530 1/20 0.36
NUDT1 P36639 1/20 0.36
PIM1 P11309 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1761836 1.00 PSMB8 (0.50) PSMB8KDM4EALDH1A1HPGDCYP3A4
SCHEMBL341252 0.75 PDE3B (0.49) ALDH1A1AURKAPARP1DAO
SCHEMBL30775064 0.69 PSMB8 (0.48) PSMB8KDM4EALDH1A1HPGDCYP3A4
SCHEMBL1002214 0.69 PSMB8 (0.48) PSMB8KDM4EALDH1A1HPGDCYP3A4
2-Mercaptobenzothiazole SCHEMBL29433968 0.67 PSMB8 (1.00) PSMB8KDM4EALDH1A1HPGDCYP3A4
2-Mercaptobenzothiazole SCHEMBL408087 0.67 PSMB8 (1.00) PSMB8KDM4EALDH1A1HPGDCYP3A4
2-Mercaptobenzothiazole SCHEMBL4268289 0.65 PSMB8 (0.95) PSMB8KDM4EALDH1A1HPGDCYP3A4
2-Mercaptobenzothiazole SCHEMBL29729650 0.65 PSMB8 (0.95) PSMB8KDM4EALDH1A1HPGDCYP3A4
2-Mercaptobenzothiazole SCHEMBL8749352 0.65 PSMB8 (0.95) PSMB8KDM4EALDH1A1HPGDCYP3A4
2-Mercaptobenzothiazole SCHEMBL5934103 0.65 PSMB8 (0.95) PSMB8KDM4EALDH1A1HPGDCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260164-B Preparation method, structural composition and application of novel 4 (3H) -quinazolinone analogue in antitumor drugs 杭州星鳌生物科技有限公司 2024-03-26 CN disclosed
CN-113717201-B (+/-) -Marinopyrole A derivative and preparation method and application thereof 植恩生物技术股份有限公司 2022-12-16 CN disclosed
WO-2022233253-A1 METHOD FOR PREPARING NEW 4(3H)-QUINAZOLINONE ANALOG, STRUCTURAL COMPOSITION THEREOF, AND USE THEREOF IN ANTITUMOR DRUGS 杭州星鳌生物科技有限公司 2022-11-10 WO disclosed
CN-115260164-A Preparation method and structural composition of novel 4 (3H) -quinazolinone analogue and application of analogue in antitumor drugs 杭州星鳌生物科技有限公司 2022-11-01 CN disclosed