SCHEMBL29968012

SCHEMBL29968012

Cc1nc2c(-c3ccc(C4=CCCCC4)cc3)cccc2n1Cc1ccc(C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.46
DCTPP1 Q9H773 1/20 0.46
PPARG P37231 7/20 0.44
PTAFR P25105 1/20 0.41
P2RX3 P56373 2/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
THRB P10828 1/20 0.40
NR4A1 P22736 1/20 0.40
APEX1 P27695 1/20 0.40
APOBEC3A P31941 1/20 0.40
RECQL P46063 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29968167 0.92 NR1H4 (0.44) NR1H4DCTPP1PPARGP2RX3
SCHEMBL29967953 0.92 PLA2G10 (0.41) NR1H4DCTPP1PPARGP2RX3KMT2A
SCHEMBL29968184 0.90 PPARG (0.43) NR1H4PPARGP2RX3ALDH1A1
SCHEMBL29968278 0.90 PPARG (0.49) NR1H4PPARGAGTR1AGTR2
SCHEMBL29967971 0.90 PPARG (0.42) DCTPP1PPARGPTAFRP2RX3AGTR1
SCHEMBL29967498 0.89 NR1H4 (0.44) NR1H4PPARGP2RX3HDAC1HDAC6
SCHEMBL29967991 0.88 PPARG (0.58) PPARGAGTR1AGTR2
SCHEMBL29968198 0.88 DCTPP1 (0.42) DCTPP1PPARGP2RX3AGTR1AGTR2
SCHEMBL29967925 0.88 PPARG (0.49) NR1H4PPARGAGTR1AGTR2
SCHEMBL29967688 0.86 CNR2 (0.38) PPARGP2RX3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed