SCHEMBL29967953

SCHEMBL29967953

Cc1nc2c(-c3ccc(C4=CCCCC4)cc3)cccc2n1Cc1cccc(C(=O)O)c1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PLA2G10 O15496 1/20 0.41
PPARG P37231 5/20 0.41
DCTPP1 Q9H773 1/20 0.40
FABP4 P15090 1/20 0.40
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
HIF1A Q16665 1/20 0.39
P2RX3 P56373 1/20 0.39
FOLH1 Q04609 1/20 0.39
CCR2 P41597 1/20 0.39
KMT2A Q03164 1/20 0.39
NR1H4 Q96RI1 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29968012 0.92 NR1H4 (0.46) PPARGDCTPP1HIF1AP2RX3KMT2A
SCHEMBL29967830 0.91 PLA2G10 (0.42) PLA2G10PPARGFABP4CYP2D6CYP2C9
SCHEMBL29967574 0.91 PPARG (0.41) PLA2G10PPARGFABP4CYP2D6CYP2C9
SCHEMBL29968086 0.91 PPARG (0.45) PLA2G10PPARG
SCHEMBL29967912 0.89 P2RX3 (0.39) PPARGDCTPP1P2RX3
SCHEMBL29967971 0.86 PPARG (0.42) PPARGDCTPP1P2RX3
SCHEMBL29967938 0.84 PPARG (0.42) PPARGP2RX3NR1H4
SCHEMBL29968167 0.84 NR1H4 (0.44) PPARGDCTPP1P2RX3NR1H4
SCHEMBL29967688 0.83 CNR2 (0.38) PPARGP2RX3
SCHEMBL29968198 0.83 DCTPP1 (0.42) PPARGDCTPP1P2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed