SCHEMBL29968169

SCHEMBL29968169

O=C(O)c1ccc(Cc2nc3c(-c4ccc(C5=CCCCC5)cc4)cccc3n2CCCO)cc1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 3/20 0.37
PPARG P37231 6/20 0.36
BRD4 O60885 1/20 0.35
CREBBP Q92793 1/20 0.35
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
JAK3 P52333 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
ACMSD Q8TDX5 1/20 0.33
PIN1 Q13526 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29968417 0.91 CNR2 (0.41) NR1H4PPARGBRD4CREBBP
SCHEMBL29967925 0.84 PPARG (0.49) NR1H4PPARG
SCHEMBL29968278 0.83 PPARG (0.49) NR1H4PPARG
SCHEMBL29967901 0.81 AGTR1 (0.56) PPARG
SCHEMBL29968167 0.81 NR1H4 (0.44) NR1H4PPARGPIN1
SCHEMBL29968012 0.81 NR1H4 (0.46) NR1H4PPARGHDAC1
SCHEMBL29967991 0.80 PPARG (0.58) PPARG
SCHEMBL29968184 0.79 PPARG (0.43) NR1H4PPARGPIN1
SCHEMBL29968438 0.79 TSHR (0.37) PPARG
SCHEMBL29967894 0.79 PPARG (0.46) PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed