SCHEMBL29968296

SCHEMBL29968296

Cc1nc2c(-c3ccc(C4=CCCCC4)cc3)cccc2n1Cc1ccccc1C#N

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.39
PIK3C2B O00750 1/20 0.38
MAPK1 P28482 1/20 0.37
ALOX5AP P20292 1/20 0.37
C5AR1 P21730 1/20 0.36
ALDH1A1 P00352 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
CNR2 P34972 1/20 0.35
DPP4 P27487 3/20 0.35
GRIN1 Q05586 2/20 0.35
GRIN2B Q13224 2/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 2/20 0.35
NPC1 O15118 1/20 0.34
GALR3 O60755 1/20 0.34
NR2F2 P24468 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29968268 0.85 KDM4E (0.43) PPARGPIK3C2BMAPK1ALOX5APALDH1A1
SCHEMBL29967780 0.82 PPARG (0.45) PPARGPIK3C2BALDH1A1
SCHEMBL29968433 0.82 CYP19A1 (0.39) PPARGPIK3C2BCNR2
SCHEMBL29968198 0.79 DCTPP1 (0.42) PPARGGALR3NR2F2RAB9A
SCHEMBL29968232 0.79 PDE10A (0.40) PPARGGALR3NR2F2RAB9A
SCHEMBL29968438 0.78 TSHR (0.37) PPARGALDH1A1NPSR1CNR2LMNA
SCHEMBL29968901 0.77 DCTPP1 (0.53) MAPK1ALDH1A1NPSR1CNR2LMNA
SCHEMBL29967688 0.77 CNR2 (0.38) PPARGCNR2
SCHEMBL29967971 0.76 PPARG (0.42) PPARG
SCHEMBL29968012 0.76 NR1H4 (0.46) PPARGALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed