SCHEMBL29968232

SCHEMBL29968232

Cc1nc2c(-c3ccc(C4=CCCCC4)cc3)cccc2n1Cc1ccncc1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.40
DCTPP1 Q9H773 1/20 0.39
AGTR1 P30556 2/20 0.37
AGTR2 P50052 2/20 0.37
HTR6 P50406 2/20 0.37
GALR3 O60755 2/20 0.37
NR2F2 P24468 2/20 0.37
RAB9A P51151 1/20 0.37
PPARG P37231 1/20 0.37
TNF P01375 1/20 0.36
EDNRA P25101 1/20 0.36
P2RX3 P56373 2/20 0.36
KCNK13 Q9HB14 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29968198 0.89 DCTPP1 (0.42) PDE10ADCTPP1AGTR1AGTR2GALR3
SCHEMBL29968901 0.88 DCTPP1 (0.53) PDE10ADCTPP1
SCHEMBL29968012 0.86 NR1H4 (0.46) DCTPP1AGTR1AGTR2PPARGP2RX3
SCHEMBL29967971 0.86 PPARG (0.42) DCTPP1AGTR1AGTR2PPARGP2RX3
SCHEMBL29968438 0.82 TSHR (0.37) PPARGP2RX3
SCHEMBL29967912 0.81 P2RX3 (0.39) DCTPP1PPARGP2RX3
SCHEMBL29967953 0.81 PLA2G10 (0.41) DCTPP1PPARGP2RX3
SCHEMBL29968268 0.81 KDM4E (0.43) PDE10AGALR3NR2F2RAB9APPARG
SCHEMBL29967688 0.81 CNR2 (0.38) PPARGP2RX3
SCHEMBL29967938 0.81 PPARG (0.42) AGTR1AGTR2PPARGP2RX3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed