SCHEMBL29976235

SCHEMBL29976235

COc1ccc(C(C)=O)c(N)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.65
HPGD P15428 5/20 0.65
CYP3A4 P08684 3/20 0.65
MAPK1 P28482 1/20 0.65
MAPT P10636 5/20 0.53
KMT2A Q03164 4/20 0.53
MEN1 O00255 3/20 0.53
KDM4E B2RXH2 3/20 0.53
GAA P10253 3/20 0.53
THRB P10828 2/20 0.53
RECQL P46063 1/20 0.53
BLM P54132 1/20 0.53
MCL1 Q07820 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
RAB9A P51151 2/20 0.52
NPC1 O15118 2/20 0.52
MAOB P27338 1/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2C19 P33261 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL312677 1.00 ALDH1A1 (0.65) ALDH1A1HPGDCYP3A4MAPK1MAPT
Hydrochloric Acid SCHEMBL30735974 0.98 ALDH1A1 (0.62) ALDH1A1HPGDCYP3A4MAPK1MAPT
Hydrochloric Acid SCHEMBL354001 0.98 ALDH1A1 (0.62) ALDH1A1HPGDCYP3A4MAPK1MAPT
SCHEMBL9929149 0.86 NPC1 (0.63) ALDH1A1HPGDCYP3A4MAPK1MAPT
SCHEMBL148855 0.85 ALDH1A1 (0.53) ALDH1A1HPGDCYP3A4MAPK1MAPT
SCHEMBL147211 0.85 SMN1; SMN2 (0.54) ALDH1A1HPGDCYP3A4MAPK1MAPT
SCHEMBL29923727 0.85 ALDH1A1 (0.59) ALDH1A1HPGDCYP3A4MAPK1MAPT
SCHEMBL632502 0.85 ALDH1A1 (0.59) ALDH1A1HPGDCYP3A4MAPK1MAPT
Hydrochloric Acid SCHEMBL30735953 0.83 ALDH1A1 (0.58) ALDH1A1HPGDCYP3A4MAPK1MAPT
SCHEMBL858839 0.83 ALDH1A1 (0.66) ALDH1A1HPGDCYP3A4MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118324761-A USP inhibitor, preparation method and application thereof 北京华森英诺生物科技有限公司 2024-07-12 CN disclosed
WO-2024003535-A2 COMPOUNDS UNIVERSITY OF DUNDEE (GB) 2024-01-04 WO disclosed
CN-115403558-A Aromatic heterocyclic compound with antitumor activity and preparation method and application thereof 河南真实生物科技有限公司 2022-11-29 CN disclosed