SCHEMBL29985287

SCHEMBL29985287

O=C(O)c1c[nH]c(=O)cc1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.45
KDM3B Q7LBC6 1/20 0.45
DYRK1A Q13627 1/20 0.45
F7 P08709 1/20 0.41
F3 P13726 1/20 0.41
CSNK2A2 P19784 3/20 0.41
CSNK2B P67870 3/20 0.41
CSNK2A1 P68400 3/20 0.41
ALDH1A1 P00352 3/20 0.40
ALOX15 P16050 1/20 0.40
ADRA1A P35348 1/20 0.40
KMT2A Q03164 2/20 0.39
NAPRT Q6XQN6 1/20 0.39
NOTUM Q6P988 2/20 0.38
CYP1A2 P05177 2/20 0.38
MEN1 O00255 1/20 0.38
HPGD P15428 1/20 0.38
ALOX12 P18054 1/20 0.38
HSD17B10 Q99714 2/20 0.37
CDC25A P30304 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1658942 0.82 ADRA1A (0.52) KDM4EKDM3BDYRK1AF7F3
SCHEMBL29799903 0.80 KDM4E (0.41) KDM4EKDM3BDYRK1AF7F3
SCHEMBL21713969 0.80 NOTUM (0.54) KDM4EKDM3BDYRK1ACSNK2A1ALDH1A1
SCHEMBL11322639 0.80 NOTUM (0.54) KDM4EKDM3BDYRK1AF7F3
SCHEMBL2336413 0.80 LCK (0.41) KDM4EKDM3BDYRK1AALDH1A1ALOX15
SCHEMBL29857063 0.80 DYRK1A (0.50) KDM4EKDM3BDYRK1AF7F3
SCHEMBL23674857 0.77 GABRP (0.40) KDM4EKDM3BDYRK1ACSNK2A2CSNK2B
SCHEMBL20606051 0.76 ALDH1A1 (0.49) KDM4EALDH1A1HPGDHSD17B10
SCHEMBL20606533 0.76 KDM4E (0.38) KDM4EKDM3BDYRK1AF7F3
SCHEMBL19817301 0.76 PRKAB2 (0.54) KDM4EDYRK1AALDH1A1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4346815-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE Schrödinger, Inc. (US) 2024-04-10 EP disclosed
CN-117715642-A Heterocyclic compounds and methods of use 薛定谔公司 2024-03-15 CN disclosed
WO-2022251497-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE SCHRÖDINGER, INC. (US) 2022-12-01 WO disclosed