SCHEMBL2998875

SCHEMBL2998875

CCCOc1ccc(-c2sc(N)c3c2C(=O)N(CCC(=O)OC)C3=O)cc1OC

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 3/20 0.38
HSD17B10 Q99714 2/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
POLB P06746 1/20 0.37
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
PRKCZ Q05513 1/20 0.36
TP53 P04637 1/20 0.35
MDM2 Q00987 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 2/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
FPR2 P25090 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2995635 0.92 ALDH1A1 (0.42) CASP3HSD17B10HPGDTSHRKDM4E
SCHEMBL2997216 0.91 CASP3 (0.42) CASP3HSD17B10HPGDKDM4EPOLB
SCHEMBL2994385 0.89 ALDH1A1 (0.42) CASP3HSD17B10HPGDKDM4EMEN1
SCHEMBL2996891 0.86 ABCB1 (0.49) CASP3HSD17B10HPGDPRKCZALDH1A1
SCHEMBL2997644 0.84 TSHR (0.41) CASP3HSD17B10HPGDTSHRKDM4E
SCHEMBL2987999 0.81 PDE4B (0.48) POLB
SCHEMBL2995604 0.80 TSHR (0.41) CASP3HSD17B10HPGDTSHRPOLB
SCHEMBL2993145 0.76 ALDH1A1 (0.42) HPGDTSHRKDM4EMEN1KMT2A
SCHEMBL2994679 0.74 LMNA (0.44) CASP3HSD17B10HPGDTSHRKDM4E
SCHEMBL2999671 0.72 PDE4B (0.42) CASP3HSD17B10HPGDTSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100179189-A1 PYRROLINE DERIVATIVES AGAINST CELL RELEASING TUMOR NECROSIS FACTOR, PREPARATION METHODS AND USES THEREOF ZHANG HESHENG 2010-07-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100179189-A1 PYRROLINE DERIVATIVES AGAINST CELL RELEASING TUMOR NECROSIS FACTOR, PREPARATION METHODS AND USES THEREOF TNF, IL1B, NOS1 CASP3 19/4885HSD17B10 3185/4885HPGD 169/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.