SCHEMBL30002576

SCHEMBL30002576

COc1cc(F)c(N)cc1OCc1cccc2ccnc(Cl)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.39
GAA P10253 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
TDP1 Q9NUW8 1/20 0.39
DCPS Q96C86 4/20 0.38
DHFR P00374 3/20 0.38
EIF2AK3 Q9NZJ5 1/20 0.36
ALDH1A1 P00352 4/20 0.35
KMT2A Q03164 3/20 0.35
KDM4E B2RXH2 2/20 0.35
MEN1 O00255 2/20 0.35
HPGD P15428 2/20 0.35
RAB9A P51151 2/20 0.35
G6PD P11413 1/20 0.34
MPO P05164 1/20 0.34
NPC1 O15118 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892669 1.00 MAPT (0.39) MAPTGAASMN1; SMN2TDP1DCPS
SCHEMBL30002446 0.88 GAA (0.40) MAPTGAASMN1; SMN2TDP1DCPS
SCHEMBL28892136 0.88 GAA (0.40) MAPTGAASMN1; SMN2TDP1DCPS
SCHEMBL28892906 0.83 LMNA (0.41) MAPTGAASMN1; SMN2ALDH1A1KMT2A
SCHEMBL30002548 0.79 SCN1A (0.47) MAPTGAASMN1; SMN2TDP1RAB9A
SCHEMBL28892526 0.79 SCN1A (0.47) MAPTGAASMN1; SMN2TDP1RAB9A
SCHEMBL30002661 0.76 MTNR1A (0.43) KMT2AMEN1MPO
SCHEMBL30002421 0.76 MEN1 (0.47) MAPTALDH1A1KMT2AKDM4EMEN1
SCHEMBL30002031 0.75 DHFR (0.38) MAPTGAASMN1; SMN2TDP1DCPS
SCHEMBL28892709 0.75 KDM4E (0.39) SMN1; SMN2KDM4EMPOCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed