SCHEMBL28892136

SCHEMBL28892136

COc1cc(F)c(N)cc1OCc1cccc2ccnc(OC)c12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
DCPS Q96C86 4/20 0.39
DHFR P00374 3/20 0.39
TRPA1 O75762 3/20 0.37
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
RAB9A P51151 1/20 0.35
MPO P05164 1/20 0.35
PIK3CG P48736 1/20 0.34
KIT P10721 1/20 0.34
PDE10A Q9Y233 1/20 0.34
CSF1R P07333 1/20 0.34
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30002446 1.00 GAA (0.40) GAAMAPTSMN1; SMN2TDP1DCPS
SCHEMBL30002576 0.88 MAPT (0.39) GAAMAPTSMN1; SMN2TDP1DCPS
SCHEMBL28892669 0.88 MAPT (0.39) GAAMAPTSMN1; SMN2TDP1DCPS
SCHEMBL30003178 0.83 LMNA (0.42) GAAMAPTSMN1; SMN2CYP1A2CYP2D6
SCHEMBL28892568 0.83 LMNA (0.42) GAAMAPTSMN1; SMN2CYP1A2CYP2D6
SCHEMBL28892526 0.80 SCN1A (0.47) GAAMAPTSMN1; SMN2TDP1RAB9A
SCHEMBL30002548 0.80 SCN1A (0.47) GAAMAPTSMN1; SMN2TDP1RAB9A
SCHEMBL30002661 0.76 MTNR1A (0.43) MPOPDE10AKMT2AMEN1
SCHEMBL30002421 0.76 MEN1 (0.47) MAPTPDE10ACSF1RKMT2AMEN1
SCHEMBL30002031 0.76 DHFR (0.38) GAAMAPTSMN1; SMN2TDP1DCPS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed