SCHEMBL30006416

SCHEMBL30006416

O=C1c2ccccc2C(=O)N1CC#Cc1cc(Br)cc(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
DRD5 P21918 1/20 0.43
P2RY6 Q15077 1/20 0.43
PTAFR P25105 8/20 0.41
PARK7 Q99497 1/20 0.39
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP1B1 Q16678 1/20 0.35
HPGD P15428 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GALR3 O60755 1/20 0.35
GSK3B P49841 1/20 0.35
RAB9A P51151 1/20 0.34
CHRM5 P08912 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27410849 0.87 ADRA2A (0.42) ADRA2AADRA2BDRD5P2RY6PTAFR
SCHEMBL30005761 0.83 PTAFR (0.41) ADRA2AADRA2BDRD5P2RY6PTAFR
SCHEMBL30006541 0.79 RAB9A (0.48) ADRA2AADRA2BDRD5P2RY6PTAFR
SCHEMBL10422970 0.73 SMN1; SMN2 (0.48) ADRA2AADRA2BDRD5P2RY6NPSR1
SCHEMBL4943682 0.71 PTAFR (0.42) ADRA2AADRA2BDRD5P2RY6PTAFR
SCHEMBL4942400 0.68 ADRA2A (0.44) ADRA2AADRA2BDRD5P2RY6PTAFR
SCHEMBL4940343 0.68 ADRA1D (0.43) ADRA2AADRA2BDRD5P2RY6PTAFR
SCHEMBL15787798 0.67 TACR1 (0.36) PARK7MEN1KMT2AHPGDNPSR1
SCHEMBL4578025 0.66 ALDH1A1 (0.47) NPSR1
SCHEMBL15787799 0.66 MAPT (0.36) PARK7MEN1KMT2ACYP1B1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022220725-A1 LPXH INHIBITORS AS ANTI-INFECTIVE AGENTS ZAMARATSKI EDOUARD (SE) 2022-10-20 WO disclosed