SCHEMBL30006541

SCHEMBL30006541

O=C1c2ccccc2C(=O)N1CC#Cc1cccc(Br)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.48
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
DRD5 P21918 1/20 0.43
P2RY6 Q15077 1/20 0.43
PTAFR P25105 8/20 0.41
GSK3B P49841 1/20 0.39
ALDH1A1 P00352 2/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38
CA12 O43570 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27410849 0.88 ADRA2A (0.42) RAB9AADRA2AADRA2BDRD5P2RY6
SCHEMBL1894591 0.83 RAB9A (0.50) RAB9AALDH1A1SMN1; SMN2CYP1B1
SCHEMBL10422970 0.82 SMN1; SMN2 (0.48) RAB9AADRA2AADRA2BDRD5P2RY6
SCHEMBL30005761 0.82 PTAFR (0.41) RAB9AADRA2AADRA2BDRD5P2RY6
SCHEMBL8902954 0.80 RXFP1 (0.46) ADRA2AADRA2BDRD5P2RY6PTAFR
SCHEMBL8803206 0.79 MMP2 (0.53) RAB9AALDH1A1POLBSMN1; SMN2MAPK1
SCHEMBL30006416 0.79 ADRA2A (0.43) RAB9AADRA2AADRA2BDRD5P2RY6
SCHEMBL4943682 0.77 PTAFR (0.42) RAB9AADRA2AADRA2BDRD5P2RY6
SCHEMBL4940343 0.74 ADRA1D (0.43) ADRA2AADRA2BDRD5P2RY6PTAFR
SCHEMBL4947503 0.73 ADRA2A (0.39) ADRA2AADRA2BDRD5P2RY6PTAFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022220725-A1 LPXH INHIBITORS AS ANTI-INFECTIVE AGENTS ZAMARATSKI EDOUARD (SE) 2022-10-20 WO disclosed