SCHEMBL30008443

SCHEMBL30008443

CCC(=O)Oc1c(-c2ccc(F)cc2)n(C)c2c(F)cc(F)cc12

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.36
POLB P06746 2/20 0.35
APOL1 O14791 3/20 0.34
FAAH O00519 2/20 0.34
ACLY P53396 2/20 0.33
USP2 O75604 1/20 0.32
MAPK14 Q16539 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30218352 0.92 FAAH (0.35) CHRNA7SMN1; SMN2APOL1FAAHUSP2
SCHEMBL30218286 0.91 POLB (0.36) CHRNA7POLBFAAHACLYMAPK14
SCHEMBL30218349 0.90 CHRNA7 (0.36) CHRNA7POLBFAAHACLYMAPK14
SCHEMBL30218302 0.89 PARP1 (0.34) POLB
SCHEMBL30218353 0.86 SMN1; SMN2 (0.38) CHRNA7SMN1; SMN2POLBAPOL1FAAH
SCHEMBL30218351 0.81 POLB (0.37) CHRNA7POLBFAAHACLYMAPK14
SCHEMBL28863434 0.72 APOL1 (0.50) APOL1
SCHEMBL10180980 0.71 KMT2A (0.39) SMN1; SMN2POLBACLY
SCHEMBL9221170 0.66 ACLY (0.50) FAAHACLY
SCHEMBL29372421 0.66 ELANE (0.40) SMN1; SMN2ACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115867543-A Solid forms of an APOL1 inhibitor and methods of use thereof 弗特克斯药品有限公司 2023-03-28 CN disclosed
CN-115867532-A Inhibitors of APOL1 and uses thereof 弗特克斯药品有限公司 2023-03-28 CN disclosed
CN-115209894-A Method for treating APOL-1 dependent focal segmental glomerulosclerosis 弗特克斯药品有限公司 2022-10-18 CN disclosed