SCHEMBL30009696

SCHEMBL30009696

CC(C)(C)OC(=O)c1c[nH]c2cc(I)ccc12

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 9/20 0.50
GABRG2 P18507 2/20 0.47
GABRB3 P28472 2/20 0.47
GABRA5 P31644 2/20 0.47
GABRA1 P14867 1/20 0.47
GABRA3 P34903 1/20 0.47
GABRA2 P47869 1/20 0.47
CREBBP Q92793 1/20 0.43
MAPT P10636 1/20 0.41
TUBB1 Q9H4B7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4375343 0.89 GABRG2 (0.53) NR4A2GABRG2GABRB3GABRA5GABRA1
SCHEMBL1696922 0.84 NR4A2 (0.51) NR4A2CREBBPMAPTTUBB1
SCHEMBL27987692 0.84 NR4A2 (0.70) NR4A2CREBBPMAPTTUBB1
SCHEMBL31618837 0.83 NR4A2 (0.56) NR4A2GABRA1GABRA3CREBBPMAPT
SCHEMBL5507447 0.83 NR4A2 (0.72) NR4A2CREBBPMAPTTUBB1
SCHEMBL7360321 0.83 NR4A2 (0.50) NR4A2GABRG2GABRB3GABRA5GABRA1
SCHEMBL6511301 0.83 NR4A2 (0.50) NR4A2CREBBPMAPTTUBB1
SCHEMBL4780483 0.82 MAPT (0.63) NR4A2MAPTTUBB1
SCHEMBL1759575 0.81 NR4A2 (0.48) NR4A2CREBBPMAPTTUBB1
SCHEMBL1696867 0.81 TUBB1 (0.50) NR4A2CREBBPMAPTTUBB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022237813-A1 COMPOUND HAVING ALK INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 盛世泰科生物医药技术(苏州)有限公司 2022-11-17 WO disclosed