SCHEMBL300208

SCHEMBL300208

Fc1cccc(-n2c[c]cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.42
FAAH O00519 1/20 0.42
MGLL Q99685 1/20 0.42
BPTF Q12830 1/20 0.36
MAPT P10636 2/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35
TUBB4B P68371 1/20 0.35
TUBB3 Q13509 1/20 0.35
TUBB2A Q13885 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2753214 0.80
SCHEMBL27634381 0.76 COMT (0.46) FAAHMGLLALDH1A1
SCHEMBL27497687 0.76 NOTUM (0.35) MGLLMAPTALDH1A1NOTUMMEN1
SCHEMBL1896817 0.76 CYP3A4 (0.40) MGLLL3MBTL1MEN1KMT2A
SCHEMBL7536022 0.76 MAPT (0.56) KEAP1FAAHMGLLMAPTALDH1A1
SCHEMBL2750984 0.72 ALDH1A1 (0.34) ALDH1A1L3MBTL1
SCHEMBL27593451 0.70 FAAH (0.46) KEAP1FAAHMGLLMAPTALDH1A1
SCHEMBL1893443 0.69 KEAP1 (0.41) KEAP1FAAHMGLLMAPTALDH1A1
SCHEMBL12841352 0.68 KEAP1 (0.52) KEAP1FAAHMGLLMAPTALDH1A1
SCHEMBL300545 0.68 KEAP1 (0.43) KEAP1FAAHMGLLBPTFMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012004443-A8 PHENYL METHYL SULFONES WITH ANTI-INFLAMMATORY ACTIVITY AND ANTI-TUMOUR ACTIVITY UNIVERSITAT DE BARCELONA (ES) 2012-02-09 WO disclosed
WO-2012004443-A1 PHENYL METHYL SULFONES WITH ANTI-INFLAMMATORY ACTIVITY AND ANTI-TUMOUR ACTIVITY UNIVERSITAT DE BARCELONA (ES) 2012-01-12 WO disclosed