SCHEMBL300545

SCHEMBL300545

Fc1cccc(-n2[c]ccc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.43
FAAH O00519 1/20 0.43
MGLL Q99685 1/20 0.43
BPTF Q12830 1/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
PI4KA P42356 1/20 0.36
PI4K2B Q8TCG2 1/20 0.36
PI4K2A Q9BTU6 1/20 0.36
PI4KB Q9UBF8 1/20 0.36
NOTUM Q6P988 2/20 0.35
METAP2 P50579 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MPI P34949 1/20 0.35
ALOX5 P09917 1/20 0.35
ACHE P22303 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11574910 0.77 MGLL (0.44) MGLLALDH1A1MAPTNOTUMMEN1
SCHEMBL8634060 0.77 NOTUM (0.47) ALDH1A1MAPTNOTUMMEN1KMT2A
SCHEMBL27629824 0.73 PRMT6 (0.41) ALDH1A1
SCHEMBL9763868 0.70 KEAP1 (0.49) KEAP1FAAHMGLLALDH1A1POLB
SCHEMBL28036187 0.70 KEAP1 (0.41) KEAP1FAAHMGLLBPTFALDH1A1
SCHEMBL7536022 0.69 MAPT (0.56) KEAP1FAAHMGLLALDH1A1POLB
SCHEMBL300208 0.68 KEAP1 (0.42) KEAP1FAAHMGLLBPTFALDH1A1
SCHEMBL2342193 0.67 KEAP1 (0.53) KEAP1FAAHMGLLBPTFALDH1A1
SCHEMBL1975063 0.67 KEAP1 (0.45) KEAP1FAAHMGLLBPTFALDH1A1
SCHEMBL16720346 0.65 HPGDS (0.39) KEAP1FAAHMGLLBPTFALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012004443-A8 PHENYL METHYL SULFONES WITH ANTI-INFLAMMATORY ACTIVITY AND ANTI-TUMOUR ACTIVITY UNIVERSITAT DE BARCELONA (ES) 2012-02-09 WO disclosed
WO-2012004443-A1 PHENYL METHYL SULFONES WITH ANTI-INFLAMMATORY ACTIVITY AND ANTI-TUMOUR ACTIVITY UNIVERSITAT DE BARCELONA (ES) 2012-01-12 WO disclosed