SCHEMBL30061908

SCHEMBL30061908

O=[N+]([O-])c1cc(OCN2CCC2)cc(C(F)(F)F)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 4/20 0.40
LTA4H P09960 3/20 0.39
PTGS2 P35354 2/20 0.39
CHRNB4 P30926 2/20 0.38
CHRNA3 P32297 2/20 0.38
PTGS1 P23219 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP3A4 P08684 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
HIF1A Q16665 1/20 0.35
TXNRD1 Q16881 1/20 0.35
TXNRD3 Q86VQ6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30063063 0.85 LTA4H (0.56) LTA4HPTGS2PTGS1HRH3MEN1
SCHEMBL545206 0.85 LTA4H (0.56) LTA4HPTGS2PTGS1HRH3MEN1
SCHEMBL13400004 0.80 ALDH1A1 (0.42) ENPP2SMN1; SMN2ALDH1A1TDP1CYP3A4
SCHEMBL30061835 0.78 ENPP2 (0.42) ENPP2SMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL16055917 0.77 RAB9A (0.48) LTA4HPTGS2PTGS1SMN1; SMN2MEN1
SCHEMBL30697141 0.77 RAB9A (0.48) LTA4HPTGS2PTGS1SMN1; SMN2MEN1
SCHEMBL1264295 0.75 ALDH1A1 (0.41) ENPP2SMN1; SMN2ALDH1A1TDP1CYP3A4
SCHEMBL1603675 0.75 LMNA (0.49) SMN1; SMN2MEN1KMT2AALDH1A1TDP1
SCHEMBL14279323 0.75 MAPT (0.38) ENPP2SMN1; SMN2ALDH1A1TDP1CYP3A4
SCHEMBL3155181 0.75 ALDH1A1 (0.39) ENPP2SMN1; SMN2MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115340552-A Heterocyclic derivative and application thereof in medicine 四川海思科制药有限公司 2022-11-15 CN disclosed