SCHEMBL30103065

SCHEMBL30103065

COc1cccc(-c2ncc(Cn3ncc4cc(Cl)cc(C(=O)NC5CC6(CC(CC(=O)O)C6)C5)c43)cn2)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.37
MCHR1 Q99705 3/20 0.36
PTGIR P43119 1/20 0.35
PTGDR Q13258 1/20 0.35
HPGDS O60760 2/20 0.35
DRD4 P21917 2/20 0.35
ROCK2 O75116 2/20 0.35
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
DRD5 P21918 1/20 0.34
AKR1C3 P42330 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
JAK1 P23458 1/20 0.34
JAK3 P52333 1/20 0.34
FFAR4 Q5NUL3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24784548 0.92 MCHR1 (0.39) MCHR1HPGDSROCK2MEN1KMT2A
SCHEMBL30103049 0.92 MCHR1 (0.39) MCHR1HPGDSROCK2MEN1KMT2A
SCHEMBL24784585 0.91 IDH1 (0.41) IDH1MCHR1PTGIRPTGDRHPGDS
SCHEMBL24785453 0.91 CRHR1 (0.37) IDH1MCHR1ROCK2
SCHEMBL30103101 0.91 CRHR1 (0.37) IDH1MCHR1ROCK2
SCHEMBL30103091 0.91 CRHR1 (0.37) IDH1MCHR1ROCK2
SCHEMBL24785852 0.90 MCHR1 (0.34) MCHR1HPGDSROCK2FFAR4
SCHEMBL30017941 0.90 MCHR1 (0.34) MCHR1HPGDSROCK2FFAR4
SCHEMBL30018138 0.89 HPGDS (0.34) MCHR1HPGDSDRD4ROCK2HDAC1
SCHEMBL30017729 0.89 ROCK2 (0.35) MCHR1ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115448913-A Bicyclic compounds for the treatment of EP2, EP4 receptor mediated diseases 武汉人福创新药物研发中心有限公司 2022-12-09 CN disclosed