SCHEMBL30104792

SCHEMBL30104792

CCOC(=O)c1cc2cc(C(F)(F)F)ncc2n1CCNC(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.39
ADORA2A P29274 1/20 0.39
BRD4 O60885 7/20 0.38
STING1 Q86WV6 2/20 0.38
DYRK1A Q13627 1/20 0.37
MTNR1A P48039 2/20 0.37
MTNR1B P49286 2/20 0.37
KDM4E B2RXH2 2/20 0.36
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
QRFPR Q96P65 1/20 0.35
MAPT P10636 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PARG Q86W56 1/20 0.34
STK17B O94768 1/20 0.34
STK17A Q9UEE5 1/20 0.34
CACNA1H O95180 1/20 0.34
CACNA1B Q00975 1/20 0.34
CACNA1C Q13936 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29878502 0.87 ADORA3 (0.40) ADORA3ADORA2ABRD4STING1DYRK1A
SCHEMBL30104845 0.83 STING1 (0.50) BRD4STING1
SCHEMBL29153650 0.83 MTNR1A (0.42) STING1MTNR1AMTNR1BKDM4ECRHBP
SCHEMBL24640541 0.81 POLB (0.41) ADORA3ADORA2ABRD4KDM4ESMN1; SMN2
Hydrochloric Acid SCHEMBL30104789 0.81 KDM4E (0.43) KDM4ECRHBPCRHR2SMN1; SMN2QRFPR
SCHEMBL24187331 0.81 MAPT (0.39) ADORA3ADORA2AMTNR1AMTNR1BKDM4E
SCHEMBL16150685 0.80 MAPT (0.47) BRD4DYRK1AMTNR1AMTNR1BKDM4E
SCHEMBL20141699 0.79 MTNR1A (0.59) MTNR1AMTNR1BKDM4ECRHBPCRHR2
SCHEMBL30681405 0.79 KDM4E (0.37) KDM4EQRFPRMAPT
SCHEMBL27341116 0.79 HPGD (0.43) ADORA3ADORA2ABRD4STING1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117396485-A PARP7 inhibitors 轩竹生物科技股份有限公司 2024-01-12 CN disclosed
WO-2022247839-A1 PARP7 INHIBITOR 山东轩竹医药科技有限公司 2022-12-01 WO disclosed