SCHEMBL30104820

SCHEMBL30104820

Fc1c2n(c3ncc(C(F)(F)F)cc13)CCNC2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 2/20 0.35
ADRB2 P07550 1/20 0.34
NCF1 P14598 1/20 0.34
POLB P06746 1/20 0.32
HTR2C P28335 2/20 0.31
HTR3E A5X5Y0 1/20 0.31
HTR3B O95264 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTR1D P28221 1/20 0.31
HTR3A P46098 1/20 0.31
HTR3D Q70Z44 1/20 0.31
HTR3C Q8WXA8 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
MCHR1 Q99705 2/20 0.31
SCN9A Q15858 1/20 0.31
HTR2A P28223 1/20 0.31
MAPT P10636 1/20 0.31
THRB P10828 1/20 0.31
GSK3B P49841 1/20 0.31
DYRK1A Q13627 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24639703 0.86 HTR2C (0.43) ADRB1ADRB2NCF1POLBHTR2C
SCHEMBL31244671 0.83 HTR2A (0.36) ADRB1ADRB2NCF1HTR2CALDH1A1
SCHEMBL30104795 0.83 PSEN1 (0.35) ADRB1ADRB2NCF1HTR2CMCHR1
SCHEMBL30720004 0.74 PARP1 (0.39)
SCHEMBL24640292 0.73 OGA (0.35) SCN9A
SCHEMBL24640572 0.73 ADRB2 (0.38) ADRB1ADRB2NCF1POLBHTR2C
SCHEMBL24640538 0.73 HTR2C (0.42) ADRB1ADRB2NCF1POLBHTR2C
SCHEMBL24640077 0.72 NR3C1 (0.34) ALDH1A1
SCHEMBL30104783 0.69 POLB (0.32) POLBALDH1A1
SCHEMBL31244768 0.67 CCRL2 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117396485-A PARP7 inhibitors 轩竹生物科技股份有限公司 2024-01-12 CN disclosed
WO-2022247839-A1 PARP7 INHIBITOR 山东轩竹医药科技有限公司 2022-12-01 WO disclosed