SCHEMBL30108043

SCHEMBL30108043

COc1ccc2c(c1)nc(-c1ccncc1)n2-c1cc(-c2ccco2)nc(N)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.41
ADORA1 P30542 4/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
HPGD P15428 1/20 0.41
ALOX12 P18054 1/20 0.41
PTPN7 P35236 1/20 0.41
HTT P42858 1/20 0.41
RECQL P46063 1/20 0.41
RAB9A P51151 1/20 0.41
BLM P54132 1/20 0.41
KMT2A Q03164 1/20 0.41
MCL1 Q07820 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
ADORA3 P0DMS8 1/20 0.40
ADORA2B P29275 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30108063 0.87 KDM4E (0.40) ADORA2AADORA1KDM4EMEN1ALDH1A1
SCHEMBL30107952 0.86 ADORA2A (0.41) ADORA2AADORA1KDM4EALDH1A1HTT
SCHEMBL30108066 0.85 ADORA2A (0.44) ADORA2AADORA1KDM4EMEN1ALDH1A1
SCHEMBL30108049 0.85 TSHR (0.45) ADORA2AADORA1KDM4EMEN1ALDH1A1
SCHEMBL30108022 0.82 SLC6A2 (0.37) ADORA2AADORA1MAPK10
SCHEMBL30107951 0.77 PTGS1 (0.46) ADORA2AADORA1KDM4EMEN1ALDH1A1
SCHEMBL30108045 0.74 ROCK1 (0.60) ADORA2AADORA1KDM4EMEN1ALDH1A1
SCHEMBL30108062 0.73 MAPT (0.39) ADORA2AADORA1KDM4EMEN1ALDH1A1
SCHEMBL30107964 0.71 ADORA2A (0.46) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL30107942 0.70 ADORA2A (0.47) ADORA2AADORA1KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022203399-A1 ADENOSINE A2A RECEPTOR ANTAGONIST AND USE THEREOF 주식회사 스탠다임 2022-09-29 WO disclosed