SCHEMBL30108045

SCHEMBL30108045

COc1ccc2c(ccn2-c2cc(-c3ccco3)nc(N)n2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 4/20 0.60
ADORA2A P29274 3/20 0.46
ADORA1 P30542 3/20 0.46
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
ADORA2B P29275 1/20 0.45
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42
THRB P10828 1/20 0.42
HPGD P15428 1/20 0.42
ALOX12 P18054 1/20 0.42
PTPN7 P35236 1/20 0.42
HTT P42858 1/20 0.42
RECQL P46063 1/20 0.42
RAB9A P51151 1/20 0.42
BLM P54132 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30107979 0.83 CDC7 (0.45) ROCK1ADORA2AADORA1ADORA3ADORA2B
SCHEMBL30107951 0.79 PTGS1 (0.46) ADORA2AADORA1PTGS1PTGS2ADORA3
SCHEMBL12821389 0.75 ROCK1 (1.00) ROCK1
SCHEMBL30108043 0.74 ADORA2A (0.41) ADORA2AADORA1PTGS1PTGS2ADORA3
SCHEMBL30108066 0.73 ADORA2A (0.44) ADORA2AADORA1PTGS1PTGS2ADORA3
SCHEMBL30353576 0.70 ALDH1A1 (0.58) ROCK1ADORA2AADORA1PTGS1PTGS2
SCHEMBL1554000 0.69 MAPT (0.58) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL5833573 0.67 ROCK1 (0.64) ROCK1MEN1POLBMAPTRAB9A
SCHEMBL29876396 0.67 ADORA2A (0.44) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL6442516 0.66 USP2 (0.62) ADORA2AADORA1ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022203399-A1 ADENOSINE A2A RECEPTOR ANTAGONIST AND USE THEREOF 주식회사 스탠다임 2022-09-29 WO disclosed