SCHEMBL30109367

SCHEMBL30109367

COc1cc(Br)ccc1N1CCc2ccccc2C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.51
ALDH1A1 P00352 4/20 0.51
HPGD P15428 1/20 0.51
POLB P06746 1/20 0.48
ACHE P22303 1/20 0.48
GRIN2D O15399 2/20 0.48
GRIN3B O60391 2/20 0.48
GRIN1 Q05586 2/20 0.48
GRIN2A Q12879 2/20 0.48
GRIN2B Q13224 2/20 0.48
GRIN2C Q14957 2/20 0.48
GRIN3A Q8TCU5 2/20 0.48
ASIC3 Q9UHC3 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
LMNA P02545 1/20 0.47
SIGMAR1 Q99720 2/20 0.47
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
DRD4 P21917 2/20 0.43
DRD1 P21728 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10536109 0.84 MAPT (0.62) MAPTALDH1A1HPGDPOLBACHE
SCHEMBL29978754 0.84 MAPT (0.62) MAPTALDH1A1HPGDPOLBACHE
SCHEMBL27946081 0.82 MAPT (0.75) MAPTALDH1A1HPGDACHEL3MBTL1
SCHEMBL30109412 0.78 MAPT (0.53) MAPTALDH1A1HPGDGRIN2DGRIN3B
SCHEMBL2799605 0.76 DRD2 (0.60) MAPTALDH1A1HPGDACHEL3MBTL1
SCHEMBL28446030 0.75 MAPT (0.53) MAPTALDH1A1HPGDPOLBGRIN2D
SCHEMBL18155195 0.73 ALDH1A1 (0.65) MAPTALDH1A1HPGDPOLBACHE
SCHEMBL4190135 0.72 HTR6 (0.61) MAPTLMNASIGMAR1
SCHEMBL20733031 0.72 CCR5 (0.52) MAPTALDH1A1HPGDACHEMEN1
SCHEMBL28511296 0.71 DRD2 (0.54) ALDH1A1HPGDDRD4HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115557889-A 2-aryl-3, 4-dihydroisoquinoline derivative and application thereof in preparing antitumor drugs 西南交通大学 2023-01-03 CN claimed
CN-115557889-A 2-aryl-3, 4-dihydroisoquinoline derivative and application thereof in preparing antitumor drugs 西南交通大学 2023-01-03 CN disclosed