SCHEMBL30120947

SCHEMBL30120947

CCOC(=O)c1cn(-c2cc([Sn](C)(C)C)ncc2C)nc1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 8/20 0.36
NPC1 O15118 4/20 0.36
RAB9A P51151 3/20 0.36
ALOX15 P16050 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
TP53 P04637 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 6/20 0.36
MAPT P10636 2/20 0.36
TSHR P16473 2/20 0.36
HSD17B10 Q99714 2/20 0.36
JMJD6 Q6NYC1 1/20 0.36
LMNA P02545 1/20 0.36
MEN1 O00255 1/20 0.36
GLA P06280 3/20 0.36
GAA P10253 3/20 0.36
CSNK1D P48730 1/20 0.36
MAPK1 P28482 1/20 0.35
HPGD P15428 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23803823 1.00 KMT2A (0.37) KMT2AALDH1A1NPC1RAB9AALOX15
SCHEMBL23803875 0.83 NPC1 (0.40) KMT2AALDH1A1NPC1RAB9AALOX15
SCHEMBL30152297 0.83 NPC1 (0.40) KMT2AALDH1A1NPC1RAB9AALOX15
SCHEMBL15310836 0.71 KMT2A (0.43) KMT2AALDH1A1NPC1RAB9AALOX15
SCHEMBL30120818 0.71 GPR52 (0.42) KMT2AALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL23803908 0.71 GPR52 (0.42) KMT2AALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL30152262 0.71 GPR52 (0.42) KMT2AALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL26659396 0.71 NPSR1 (0.47) KMT2AALDH1A1NPC1RAB9ANPSR1
SCHEMBL17980321 0.70 NPC1 (0.49) KMT2AALDH1A1NPC1RAB9ANPSR1
SCHEMBL15051243 0.69 ALDH1A1 (0.36) KMT2AALDH1A1NPC1RAB9AALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115515681-B GPR52 modulator compounds 奈克斯拉制药英国有限公司 2024-09-03 CN disclosed
EP-4117784-A1 GPR52 MODULATOR COMPOUNDS Heptares Therapeutics Limited (GB) 2023-01-18 EP disclosed
CN-115515681-A GPR52 modulator compounds 赫普泰雅治疗有限公司 2022-12-23 CN disclosed