SCHEMBL30152297

SCHEMBL30152297

CCOC(=O)c1cn(-c2cc(Br)ncc2C)nc1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.40
KMT2A Q03164 3/20 0.40
RAB9A P51151 3/20 0.40
MEN1 O00255 2/20 0.40
LMNA P02545 2/20 0.40
ALDH1A1 P00352 6/20 0.38
ALOX15 P16050 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
TP53 P04637 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 4/20 0.37
MAPT P10636 2/20 0.37
TSHR P16473 2/20 0.37
HSD17B10 Q99714 1/20 0.37
JMJD6 Q6NYC1 1/20 0.37
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
CSNK1D P48730 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23803875 1.00 NPC1 (0.40) NPC1KMT2ARAB9AMEN1LMNA
SCHEMBL30120947 0.83 KMT2A (0.37) NPC1KMT2ARAB9AMEN1LMNA
SCHEMBL23803823 0.83 KMT2A (0.37) NPC1KMT2ARAB9AMEN1LMNA
SCHEMBL6766046 0.75 NPC1 (0.46) NPC1RAB9ALMNAALDH1A1NPSR1
SCHEMBL23803909 0.73 LMNA (0.47) NPC1KMT2ARAB9AMEN1LMNA
SCHEMBL15310836 0.73 KMT2A (0.43) NPC1KMT2ARAB9AMEN1LMNA
SCHEMBL23803908 0.73 GPR52 (0.42) NPC1KMT2ARAB9AMEN1ALDH1A1
SCHEMBL30152262 0.73 GPR52 (0.42) NPC1KMT2ARAB9AMEN1ALDH1A1
SCHEMBL30120818 0.73 GPR52 (0.42) NPC1KMT2ARAB9AMEN1ALDH1A1
SCHEMBL26005165 0.73 CA12 (0.61) NPC1KMT2ARAB9AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115515681-B GPR52 modulator compounds 奈克斯拉制药英国有限公司 2024-09-03 CN disclosed
CN-115515681-A GPR52 modulator compounds 赫普泰雅治疗有限公司 2022-12-23 CN disclosed