SCHEMBL30131399

SCHEMBL30131399

O=C(NCC(F)(F)C(F)(F)C(F)(F)F)c1ncccc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.40
EGLN2 Q96KS0 1/20 0.40
FTO Q9C0B1 1/20 0.40
NR3C1 P04150 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
CTSA P10619 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HSD17B13 Q7Z5P4 1/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37
GRM1 Q13255 1/20 0.37
TRPV1 Q8NER1 2/20 0.37
MAPK8 P45983 1/20 0.36
GAA P10253 1/20 0.36
TLR7 Q9NYK1 2/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30131356 0.92 EGLN2 (0.41) EGLN2FTONR3C1CYP1A2CYP3A4
SCHEMBL30131474 0.86 LOXL2 (0.45) EGLN2FTONR3C1CYP1A2CYP3A4
SCHEMBL30131499 0.80 EGLN2 (0.43) EGLN2FTOCTSAALDH1A1POLB
SCHEMBL30875096 0.78 RAB9A (0.46) EGLN2FTOALDH1A1HSD17B13HPGD
SCHEMBL24869259 0.76 CFTR (0.41) CA2EGLN2ALDH1A1NPC1RAB9A
SCHEMBL30875055 0.76 EGLN2 (0.44) EGLN2FTOCTSAALDH1A1POLB
SCHEMBL30131408 0.75 NPC1 (0.47) EGLN2FTOALDH1A1POLBHPGD
SCHEMBL30875025 0.74 ALDH1A1 (0.43) EGLN2FTOCTSAALDH1A1POLB
SCHEMBL29459608 0.74 POLB (0.47) EGLN2FTOPOLBHPGDNPC1
SCHEMBL31384297 0.73 P2RX7 (0.52) EGLN2FTOCTSAALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023279986-A1 SIX-MEMBERED ARYL OR HETEROARYL AMIDES, AND COMPOSITION AND USE THEREOF 贝达药业股份有限公司 2023-01-12 WO claimed
WO-2023279986-A1 SIX-MEMBERED ARYL OR HETEROARYL AMIDES, AND COMPOSITION AND USE THEREOF 贝达药业股份有限公司 2023-01-12 WO disclosed