SCHEMBL30132085

SCHEMBL30132085

NC(=O)c1cnn(-c2cccc(N)c2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.51
ALKBH2 Q6NS38 1/20 0.51
BTK Q06187 1/20 0.47
NPC1 O15118 5/20 0.46
MAP4K4 O95819 1/20 0.45
MLLT3 P42568 1/20 0.44
MLLT1 Q03111 1/20 0.44
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
RAB9A P51151 5/20 0.43
MAPT P10636 4/20 0.43
HPGD P15428 2/20 0.43
HTT P42858 2/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
MAPKAPK2 P49137 1/20 0.42
PARP1 P09874 1/20 0.41
PARP15 Q460N3 1/20 0.41
PARP10 Q53GL7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4481678 1.00 HPGDS (0.51) HPGDSALKBH2BTKNPC1MAP4K4
SCHEMBL3374557 0.88 ALKBH2 (0.69) HPGDSALKBH2NPC1MLLT3MLLT1
SCHEMBL5063087 0.87 HPGDS (0.50) HPGDSALKBH2BTKNPC1MAP4K4
SCHEMBL2190049 0.82 ALKBH2 (0.74) HPGDSALKBH2NPC1MAP4K4RAB9A
SCHEMBL10139147 0.81 MAP4K4 (0.56) HPGDSALKBH2BTKNPC1MAP4K4
SCHEMBL3107063 0.80 EPHX2 (0.64) HPGDSALKBH2BTKNPC1RAB9A
SCHEMBL30978305 0.78 BTK (0.48) HPGDSALKBH2BTKNPC1RAB9A
SCHEMBL23846557 0.77 F7 (0.54) HPGDSALKBH2BTKNPC1MAP4K4
SCHEMBL4500055 0.76 SCN9A (0.54) HPGDSALKBH2BTKNPC1MAP4K4
Isophthalic Acid SCHEMBL27862943 0.74 ALKBH2 (0.54) HPGDSALKBH2NPC1KEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4100015-A1 COMBINATION THERAPY FOR TREATING MPS1 Gain Therapeutics SA (CH) 2022-12-14 EP disclosed