SCHEMBL30145150

SCHEMBL30145150

N#Cc1ccc(C2=Nc3ccccc3Cc3ccccc32)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 3/20 0.46
RARA P10276 1/20 0.41
RARB P10826 1/20 0.41
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
RXRG P48443 1/20 0.41
HRH4 Q9H3N8 1/20 0.40
LAP3 P28838 1/20 0.36
MAOB P27338 1/20 0.36
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
IDO1 P14902 2/20 0.35
CYP11B2 P19099 3/20 0.35
FABP1 P07148 1/20 0.33
KIF11 P52732 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14507199 0.82 IDO1 (0.50) TRPA1RARARARBRXRARXRB
SCHEMBL30145190 0.80 HRH4 (0.47) TRPA1RARARARBRXRARXRB
SCHEMBL30145076 0.77 RARA (0.46) RARARARBRXRARXRBRXRG
SCHEMBL14507248 0.75 HDAC3 (0.56) TRPA1RARARARBRXRARXRB
SCHEMBL5366018 0.74 HRH4 (0.46) TRPA1HRH4LMNAMAPTIDO1
SCHEMBL7701030 0.73 NOS3 (0.45) LAP3MAOBLMNAMAPTIDO1
SCHEMBL28246117 0.72 PDK2 (0.50) TRPA1LAP3MAOBLMNAMAPT
SCHEMBL30145240 0.71 GSK3A (0.46) RARARARBRXRARXRBRXRG
SCHEMBL29234139 0.70 OPRD1 (0.37) TRPA1MAOBIDO1CYP11B2TSHR
SCHEMBL27740845 0.69 LAP3 (0.51) HRH4LAP3MAOBCYP11B2FABP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113072500-B Synthetic method of dibenzo [ b, e ] azepine compound 淮北师范大学 2023-01-20 CN disclosed