SCHEMBL30162823

SCHEMBL30162823

O=[N+]([O-])c1cc(F)c2c(cnn2C2CCCCO2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.45
CYP4F2 P78329 2/20 0.41
CYP4A11 Q02928 2/20 0.41
ALDH1A1 P00352 4/20 0.39
LMNA P02545 2/20 0.39
POLB P06746 1/20 0.39
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
CYP1A2 P05177 1/20 0.35
HPGD P15428 1/20 0.35
ATR Q13535 4/20 0.33
RAB9A P51151 2/20 0.32
NPC1 O15118 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
OPRK1 P41145 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
KMT2A Q03164 1/20 0.31
ESR1 P03372 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29218312 1.00 EGFR (0.45) EGFRCYP4F2CYP4A11ALDH1A1LMNA
SCHEMBL21198422 0.87 CYP1A2 (0.42) EGFRCYP4F2CYP4A11ALDH1A1LMNA
SCHEMBL31539789 0.84 CYP4F2 (0.46) EGFRCYP4F2CYP4A11ALDH1A1LMNA
SCHEMBL19204859 0.82 CYP4F2 (0.47) EGFRCYP4F2CYP4A11ALDH1A1LMNA
SCHEMBL19204864 0.81 CYP4F2 (0.44) EGFRCYP4F2CYP4A11ALDH1A1LMNA
SCHEMBL767235 0.81 CYP4F2 (0.44) EGFRCYP4F2CYP4A11ALDH1A1LMNA
SCHEMBL30162853 0.81 LMNA (0.48) EGFRCYP4F2CYP4A11ALDH1A1LMNA
SCHEMBL25073931 0.79 CYP4F2 (0.42) EGFRCYP4F2CYP4A11ALDH1A1LMNA
SCHEMBL5413224 0.79 RXRA (0.54) CYP4F2CYP4A11ALDH1A1LMNAPOLB
SCHEMBL21202197 0.79 ALDH1A1 (0.40) EGFRCYP4F2CYP4A11ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4377306-A1 ROCK2 INHIBITORS AND USES THEREOF President and Fellows of Harvard College (US) 2024-06-05 EP disclosed
WO-2023009475-A1 ROCK2 INHIBITORS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2023-02-02 WO disclosed