SCHEMBL3019

SCHEMBL3019

CC(OC(=O)c1ccccc1-c1ccc(CNC(CO)Cc2ccccc2)cc1)[Si](C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 1/20 0.42
PDCD1 Q15116 2/20 0.42
CD274 Q9NZQ7 2/20 0.42
BACE1 P56817 1/20 0.41
SCN1A P35498 1/20 0.41
SCN2A Q99250 1/20 0.41
SCN3A Q9NY46 1/20 0.41
BDKRB1 P46663 3/20 0.41
MAPK1 P28482 2/20 0.40
CYP3A4 P08684 1/20 0.40
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
ROCK2 O75116 3/20 0.39
ROCK1 Q13464 3/20 0.39
MME P08473 3/20 0.38
MMEL1 Q495T6 1/20 0.38
RPS6KA5 O75582 1/20 0.38
RPS6KA4 O75676 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3035 0.93 SLC6A4 (0.47) ADRB3PDCD1CD274BACE1SCN1A
SCHEMBL2721 0.85 BDKRB1 (0.39) ADRB3PDCD1CD274SCN1ASCN2A
SCHEMBL2970 0.85 BDKRB1 (0.39) ADRB3PDCD1CD274SCN1ASCN2A
SCHEMBL3020 0.83 SCN1A (0.42) ADRB3PDCD1CD274BACE1SCN1A
SCHEMBL2126 0.80 SCN1A (0.48) SCN1ASCN2ASCN3ABDKRB1LTB4R2
SCHEMBL1639 0.80 SLC6A4 (0.48) PDCD1CD274SCN1ASCN2ASCN3A
SCHEMBL3201 0.78 SCN1A (0.49) SCN1ASCN2ASCN3ABDKRB1LTB4R2
SCHEMBL3036 0.77 SLC6A4 (0.46) PDCD1CD274SCN1ASCN2ASCN3A
SCHEMBL2301 0.75 SCN1A (0.47) SCN1ASCN2ASCN3AMAPK1
SCHEMBL28653629 0.73 SIGMAR1 (0.51) BACE1MAPK1CYP3A4ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0443983-B1 Acyl compounds CIBA GEIGY AG (CH) 1996-02-28 EP disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed