SCHEMBL3035

SCHEMBL3035

CC(OC(=O)c1ccccc1-c1ccc(CNC(CO)Cc2ccc(F)cc2)cc1)[Si](C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.47
SLC6A3 Q01959 1/20 0.47
BDKRB1 P46663 5/20 0.39
ADRB3 P13945 1/20 0.39
PDCD1 Q15116 2/20 0.38
CD274 Q9NZQ7 2/20 0.38
SCN1A P35498 1/20 0.37
SCN2A Q99250 1/20 0.37
SCN3A Q9NY46 1/20 0.37
MME P08473 6/20 0.37
MMEL1 Q495T6 1/20 0.37
BRS3 P32247 1/20 0.36
BACE1 P56817 1/20 0.36
ACE P12821 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3019 0.93 ADRB3 (0.42) BDKRB1ADRB3PDCD1CD274SCN1A
SCHEMBL1639 0.87 SLC6A4 (0.48) SLC6A4SLC6A3BDKRB1PDCD1CD274
SCHEMBL3036 0.84 SLC6A4 (0.46) SLC6A4SLC6A3BDKRB1PDCD1CD274
SCHEMBL2721 0.83 BDKRB1 (0.39) BDKRB1ADRB3PDCD1CD274SCN1A
SCHEMBL2970 0.83 BDKRB1 (0.39) BDKRB1ADRB3PDCD1CD274SCN1A
SCHEMBL2126 0.78 SCN1A (0.48) SLC6A4SLC6A3BDKRB1SCN1ASCN2A
SCHEMBL3020 0.77 SCN1A (0.42) BDKRB1ADRB3PDCD1CD274SCN1A
SCHEMBL3201 0.76 SCN1A (0.49) SLC6A4SLC6A3BDKRB1SCN1ASCN2A
SCHEMBL2746 0.73 AGTR1 (0.53) SLC6A4SLC6A3
SCHEMBL2301 0.73 SCN1A (0.47) SLC6A4SLC6A3SCN1ASCN2ASCN3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965592-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1999-10-12 US disclosed
EP-0443983-B1 Acyl compounds CIBA GEIGY AG (CH) 1996-02-28 EP disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed