SCHEMBL3020

SCHEMBL3020

C[Si](C)(C)CCOC(=O)c1ccccc1-c1ccc(CNC(CO)Cc2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 2/20 0.42
SCN2A Q99250 2/20 0.42
SCN3A Q9NY46 2/20 0.42
PDCD1 Q15116 2/20 0.41
CD274 Q9NZQ7 2/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNA4 P43681 1/20 0.41
LTB4R2 Q9NPC1 1/20 0.39
BACE1 P56817 1/20 0.39
BDKRB1 P46663 4/20 0.38
ROCK2 O75116 3/20 0.38
ROCK1 Q13464 3/20 0.38
ADRB3 P13945 1/20 0.38
MAPK1 P28482 2/20 0.38
RPS6KA5 O75582 1/20 0.38
RPS6KA4 O75676 1/20 0.38
PRKACA P17612 1/20 0.38
GSK3A P49840 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3036 0.93 SLC6A4 (0.46) SCN1ASCN2ASCN3APDCD1CD274
SCHEMBL2722 0.85 BDKRB1 (0.36) SCN1ASCN2ASCN3APDCD1CD274
SCHEMBL2971 0.85 BDKRB1 (0.36) SCN1ASCN2ASCN3APDCD1CD274
SCHEMBL3019 0.83 ADRB3 (0.42) SCN1ASCN2ASCN3APDCD1CD274
SCHEMBL2127 0.79 SCN1A (0.50) SCN1ASCN2ASCN3ACHRNB2CHRNB4
SCHEMBL3202 0.77 SCN1A (0.51) SCN1ASCN2ASCN3ACHRNB2CHRNB4
SCHEMBL3035 0.77 SLC6A4 (0.47) SCN1ASCN2ASCN3APDCD1CD274
SCHEMBL2302 0.75 SCN1A (0.51) SCN1ASCN2ASCN3ACHRNB2CHRNB4
SCHEMBL1615 0.72 SCN1A (0.51) SCN1ASCN2ASCN3ACHRNB2CHRNB4
SCHEMBL28653631 0.72 SIGMAR1 (0.51) BACE1ROCK2ROCK1MAPK1RPS6KA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0443983-B1 Acyl compounds CIBA GEIGY AG (CH) 1996-02-28 EP disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed