SCHEMBL30201463

SCHEMBL30201463

O=C(O)c1ccc2ccn(-c3ccc(F)cc3)c2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.60
MGLL Q99685 3/20 0.45
KCNH2 Q12809 1/20 0.44
BCL2L1 Q07817 1/20 0.43
BAD Q92934 1/20 0.43
F2 P00734 2/20 0.42
F10 P00742 2/20 0.42
PRSS1 P07477 2/20 0.42
FGFR1 P11362 1/20 0.41
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 3/20 0.40
MAPT P10636 2/20 0.40
HPGD P15428 2/20 0.40
NPC1 O15118 1/20 0.40
TSHR P16473 1/20 0.40
ALOX12 P18054 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP1A2 P05177 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL121755 0.88 MGLL (0.56) SCN9AMGLLKCNH2BCL2L1BAD
SCHEMBL24950460 0.86 FGFR1 (0.55) SCN9AF2F10PRSS1FGFR1
SCHEMBL30201454 0.86 FGFR1 (0.55) SCN9AF2F10PRSS1FGFR1
SCHEMBL29280306 0.85 SRD5A2 (0.49) SCN9AMGLLKCNH2F2F10
SCHEMBL18002655 0.83 KDM4E (0.54) SCN9AKCNH2KDM4EALDH1A1MAPT
SCHEMBL30201485 0.82 SCN9A (0.48) SCN9AF2F10PRSS1FGFR1
SCHEMBL2610323 0.78 KCNH2 (0.48) SCN9AMGLLKCNH2KDM4EALDH1A1
SCHEMBL2610321 0.78 KCNH2 (0.47) SCN9AMGLLKCNH2KDM4EALDH1A1
SCHEMBL28311684 0.77 SCN9A (0.44) SCN9AF2F10PRSS1FGFR1
SCHEMBL6840200 0.76 RXRA (0.47) SCN9AMGLLKCNH2FGFR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117729914-A Serotonin 5-HT2B inhibiting compounds 硕腾服务有限责任公司 2024-03-19 CN disclosed
WO-2023009330-A1 SEROTONIN 5-HT2B INHIBITORY COMPOUNDS ZOETIS SERVICES LLC (US) 2023-02-02 WO disclosed