SCHEMBL30205490

SCHEMBL30205490

COc1ccc(CS(=O)(=O)c2ccc(N(C)C)c([N+](=O)[O-])c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
KDM4E B2RXH2 1/20 0.54
HTT P42858 1/20 0.54
TXNRD1 Q16881 7/20 0.53
POLB P06746 2/20 0.51
MCOLN3 Q8TDD5 1/20 0.51
CYP19A1 P11511 1/20 0.46
RAB9A P51151 2/20 0.44
GALR3 O60755 1/20 0.44
NR2F2 P24468 1/20 0.44
MAPT P10636 2/20 0.43
LMNA P02545 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
GAA P10253 1/20 0.42
PKM P14618 1/20 0.42
MAPK1 P28482 1/20 0.42
ALDH3A1 P30838 1/20 0.42
HCAR3 P49019 1/20 0.42
KEAP1 Q14145 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30205334 0.85 ALDH1A1 (0.57) ALDH1A1KDM4EHTTTXNRD1CYP19A1
SCHEMBL7533291 0.82 TXNRD1 (0.58) ALDH1A1TXNRD1MAPTLMNAMAPK1
SCHEMBL7540192 0.82 TXNRD1 (0.55) ALDH1A1HTTTXNRD1CYP19A1RAB9A
SCHEMBL3991397 0.78 POLB (0.62) ALDH1A1KDM4EHTTPOLBMCOLN3
SCHEMBL30205148 0.77 ALDH1A1 (0.53) ALDH1A1KDM4EHTTTXNRD1POLB
SCHEMBL7540268 0.73 VCAM1 (0.58) ALDH1A1TXNRD1
SCHEMBL29029059 0.71 ALDH1A1 (0.50) ALDH1A1KDM4EHTTPOLBMCOLN3
SCHEMBL10060156 0.71 ALDH1A1 (0.71) ALDH1A1KDM4EHTTPOLBMCOLN3
SCHEMBL6517136 0.71 ALDH1A1 (0.71) ALDH1A1KDM4EHTTPOLBMCOLN3
SCHEMBL29029071 0.71 ALDH1A1 (0.49) ALDH1A1KDM4EHTTPOLBMCOLN3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115710251-A Myeloid differentiation factor 88 inhibitor and preparation method and application thereof 杭州医学院 2023-02-24 CN claimed
CN-115710251-B Medullary differentiation factor 88 inhibitor and preparation method and application thereof 杭州医学院 2024-05-28 CN disclosed
CN-115710251-A Myeloid differentiation factor 88 inhibitor and preparation method and application thereof 杭州医学院 2023-02-24 CN disclosed